| 英文名稱 | Rupatadine Fumarate | UR-12592 Fumarate |
|---|---|
| 中文名稱 | 富馬酸盧帕他定 |
| CAS號 | 182349-12-8 |
| 分子式 | C26H26ClN3·C4H4O4 |
| 分子量 | 532.03 | 415.97(free) |
| 外觀 | White to off-white powder |
| 儲存條件 | 4°C, sealed storage, away from moisture |
| 英文名稱 | Rupatadine Fumarate | UR-12592 Fumarate |
|---|---|
| 中文名稱 | 富馬酸盧帕他定 |
| CAS號 | 182349-12-8 |
| 分子式 | C26H26ClN3·C4H4O4 |
| 分子量 | 532.03 | 415.97(free) |
| 外觀 | White to off-white powder |
| 儲存條件 | 4°C, sealed storage, away from moisture |
Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively.
PMID: 8996188
Rupatadine protects against pulmonary fibrosis by attenuating PAF-mediated senescence in rodents.
PMID: 23869224 PMCID: PMC3711902 DOI: 10.1371/journal.pone.0068631
PMID: 10959557 DOI: 10.1007/PL00000216